2. Signaling Pathways
  3. Metabolic Enzyme/Protease
  4. Drug Metabolite

Drug Metabolite

Drug Metabolite

Related Products

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Drug metabolite results when a drug is metabolized into a modified form which continues to produce effects. Drug metabolism redox reactions such as heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations can yield active metabolites, and in rare cases even conjugation reactions can yield an active metabolite.

Cat. No. Product Name Effect Purity Chemical Structure
  • HY-15405R
    Teriflunomide (Standard)
    Teriflunomide (Standard) is the analytical standard of Teriflunomide. This product is intended for research and analytical applications. Teriflunomide is the active metabolite of leflunomide, an approved therapy for rheumatoid arthritis. It inhibits pyrimidine synthesis and therefore potently decreases T cell and B cell proliferation.
    Teriflunomide (Standard)
  • HY-114547R
    PD 109488 (Standard)
    PD 109488 (Standard) is the analytical standard of PD 109488. This product is intended for research and analytical applications. PD 109488 is a quinapril diketopiperazine metabolite.
    PD 109488 (Standard)
  • HY-135394R
    3-Desacetyl Cefotaxime lactone (Standard)
    3-Desacetyl Cefotaxime lactone (Standard) is the analytical standard of 3-Desacetyl Cefotaxime lactone. This product is intended for research and analytical applications. 3-Desacetyl Cefotaxime lactone is the active metabolite of Cefotaxime. Cefotaxime sodium salt is a third-generation cephalosporin antibiotic.
    3-Desacetyl Cefotaxime lactone (Standard)
  • HY-133694R
    2-Aminoflubendazole (Standard)
    2-Aminoflubendazole (Standard) is the analytical standard of 2-Aminoflubendazole. This product is intended for research and analytical applications. 2-Aminoflubendazole is the metabolite of Benzimidazoles. Benzimidazoles (BZ) are a class of agents with activities against fungi, protozoa, and helminthes.
    2-Aminoflubendazole (Standard)
  • HY-113095R
    γ-CEHC (Standard)
    Ftivazide (Standard) is the analytical standard of Ftivazide. This product is intended for research and analytical applications. Ftivazide has anti-tuberculosis activity.
    γ-CEHC (Standard)
  • HY-W016221R
    6-Hydroxy Chlorzoxazone (Standard)
    6-Hydroxy Chlorzoxazone (Standard) is the analytical standard of 6-Hydroxy Chlorzoxazone. This product is intended for research and analytical applications. 6-Hydroxy Chlorzoxazone is a metabolite of Chlorzoxazone (HY-B1462). Chlorzoxazone is a centrally acting muscle relaxant used to treat muscle spasm and the resulting pain or discomfort.
    6-Hydroxy Chlorzoxazone (Standard)
  • HY-126129R
    Desacetylcefotaxime (Standard)
    Desacetylcefotaxime (Standard) is the analytical standard of Desacetylcefotaxime. This product is intended for research and analytical applications. Desacetylcefotaxime, the in vivo metabolite of Cefotaxime (CTX), possesses significant in vitro antimicrobial activity similar to the parent compound against a variety of aerobic and anaerobic bacteria.
    Desacetylcefotaxime (Standard)
  • HY-N8483
    Eprinomectin B1a
    Eprinomectin B1a is a Eprinomectin (HY-12643) metabolite (an antiparasitic compound).
    Eprinomectin B1a
  • HY-G0001
    Lurasidone metabolite 14283
    Lurasidone metabolite 14283 is an active metabolite of lurasidone (HY-B0032A) and can be used in antipsychotic research.
    Lurasidone metabolite 14283
  • HY-W750297
    p,p'-DDD-13C12
    p,p'-DDD-13C12 is 13C labeled p,p'-DDD. p,p'-DDD is a major metabolite of p,p'-DDT. p,p'-DDD occurs in the feces and livers of rats, that are given p,p'-DDT by stomach tube, but not of rats injected intraperitoneally with p,p'-DDT.
    p,p'-DDD-<sup>13</sup>C<sub>12</sub>
  • HY-124414A
    4'-Hydroxytamoxifen TFA
    		99.43%
    4'-Hydroxytamoxifen TFA is a salt form of a metabolite of Tamoxifen. 4'-Hydroxytamoxifen TFA has a higher affinity for ER than Tamoxifen. 4'-Hydroxytamoxifen TFA induces non-apoptotic cytotoxicity in human endometrial adenocarcinoma cells.
    4'-Hydroxytamoxifen TFA
  • HY-146269
    11-Desethyl Irinotecan
    11-Desethyl Irinotecan is a camptothecin (CPT) analog and one of the metabolites of irinotecan. It is promising for cancer research.
    11-Desethyl Irinotecan
  • HY-125850R
    Berberrubine chloride (Standard)
    Berberrubine (chloride) (Standard) is the analytical standard of Berberrubine (chloride). This product is intended for research and analytical applications. Berberrubine chloride is an orally active metabolite of berberine. Berberrubine chloride alleviates mucosal lesions and inflammation in mouse colitis models. Berberrubine chloride has anti-inflammatory, anti-tumor, and antiviral activities.
    Berberrubine chloride (Standard)
  • HY-W410706
    1-Salicylate glucuronide
    1-Salicylate glucuronide is a metabolite of Salicylic acid (HY-B0167) and Aspirin (HY-14654).
    1-Salicylate glucuronide
  • HY-15852
    THRX-195518
    THRX-195518 is the major metabolite of Revefenacin (HY-15851), a lung-selective and long-acting muscarinic antagonist. THRX-195518 can be utilized in research related to chronic obstructive pulmonary disease.
    THRX-195518
  • HY-W086896R
    α-Demethylnaproxen (Standard)
    α-Demethylnaproxen (Standard) is the analytical standard of α-Demethylnaproxen. This product is intended for research and analytical applications. α-Demethylnaproxen is the major metabolite of Nabumetone (HY-B0559), Nabumetone is an orally active COX-2 inhibitor with anti-inflammatory activity.
    α-Demethylnaproxen (Standard)
  • HY-G0012S
    Monohydroxy Netupitant-d6
    Monohydroxy Netupitant-d6 is the deuterium labeled Monohydroxy Netupitant, which is a metabolite of Netupitant.
    Monohydroxy Netupitant-d<sub>6</sub>
  • HY-W104076
    2-Amino-2'-fluoro-5-nitrobenzophenone
    		Control 99.88%
    2-Amino-2'-fluoro-5-nitrobenzophenone is a precursor in the synthesis of benzodiazepines. 2-Amino-2'-fluoro-5-nitrobenzophenone is also an acid hydrolysis product of Flunitrazepam.
    2-Amino-2'-fluoro-5-nitrobenzophenone
  • HY-12388S1
    N-Desmethyl clomipramine-d6
    N-Desmethyl clomipramine-d6 (Desmethylclomipramine-d6) is deuterium labeled N-Desmethyl clomipramine. Desmethylclomipramine (Norclomipramine) is a metabolite of Clomipramine (HY-B0457A) and can be used for neurological research.
    N-Desmethyl clomipramine-d<sub>6</sub>
  • HY-W742417
    Tazarotenic acid-d8
    Tazarotenic acid-d8 (AGN 190299-d8) is the deuterium labeled Tazarotenic acid (HY-101108). Tazarotenic acid is the metabolite of Tazarotene (HY-15388).
    Tazarotenic acid-d<sub>8</sub>
Cat. No. Product Name / Synonyms Application Reactivity